PIDA-mediated oxidative C-C bond formation: novel synthesis of indoles from N-aryl enamines.
PIDA-mediated oxidative C-C bond formation: novel synthesis of indoles from N-aryl enamines.
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DOI：
10.1021/ol900576a
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发表时间：
2009-05
期刊：
影响因子：
5.2
通讯作者：
Wenquan Yu;Yunfei Du;K. Zhao
中科院分区：
文献类型：
--
作者：
Wenquan Yu;Yunfei Du;K. Zhao
通过 PIDA 介导的氧化碳-碳键形成，由 N-芳基烯胺合成了多种功能化吲哚。该反应的特点包括底物2的制备容易、官能团耐受性好、反应条件温和、不含过渡金属等。
A variety of functionalized indoles were synthesized from N-aryl enamines via PIDA-mediated oxidative carbon-carbon bond formation. The features of the present reaction include facilitative preparation of substrates 2, good functional group tolerance, and mild reaction conditions without transition metals.