Palladium-catalyzed arylation of electron-rich heterocycles with aryl chlorides
Palladium-catalyzed arylation of electron-rich heterocycles with aryl chlorides
复制标题
DOI：
10.1021/ol0702324
复制
发表时间：
2007-04-12
期刊：
影响因子：
5.2
通讯作者：
Daugulis, Olafs
中科院分区：
文献类型：
--
作者：
Chiong, Hendrich A.;Daugulis, Olafs
钯催化的C-H激活：现在可以将廉价的芳基氯化物用于各种富含电子的杂环的芳基化。该反应成功的关键是使用庞大的，富含电子的磷酸配体。不需要铜添加剂。
Palladium-catalyzed C-H activation: cheap aryl chlorides can now be used for the arylation of a wide variety of electron-rich heterocycles. The key to the success of this reaction is the use of a bulky, electron-rich phosphine ligand. No copper additives are needed.