Compounds structurally related to tamoxifen as openers of large-conductance calcium-activated K+ channel.

Compounds structurally related to tamoxifen as openers of large-conductance calcium-activated K+ channel.
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结构上与他莫昔芬相关的化合物作为大电导钙激活 K 通道的开启剂。

DOI:
10.1248/cpb.53.1372
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发表时间:
2005
影响因子:
1.7
通讯作者:
T. Ohwada
T. Ohwada
中科院分区:
医学4区
文献类型:
--
作者:
Yu Sha;T. Tashima;Yumi Mochizuki;Yoshimi Toriumi;S. Adachi;Taro Nonomura;M. Cheng;T. Ohwada

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我们发现多种含有他莫昔芬部分结构的化合物显示出作为大电导钙活化K+通道(BK通道)的化学调节剂的活性。
We found that a variety of compounds containing partial structures of tamoxifen showed activity as chemical modulators of large-conductance calcium-activated K+ channels (BK channels).
DOI: 10.1073/pnas.93.17.9200
发表时间: 1996-08-20
影响因子: 11.1
作者:
TsengCrank, J;Godinot, N;Reinhart, PH
通讯作者: Reinhart, PH