Directed ortho lithiation of N-alkylphenylaziridines
Directed ortho lithiation of N-alkylphenylaziridines
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DOI：
10.1021/ol051412l
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发表时间：
2005-08-18
期刊：
影响因子：
5.2
通讯作者：
Musio, B
中科院分区：
文献类型：
--
作者：
Capriati, V;Florio, S;Musio, B
[GRAPHICS]The ortho lithiation-trapping sequence of phenylaziridines is described. This methodology, which counts on the ability of the aziridino group to act as a directed metalation group (DMG), provides an easy access to functionalized arylaziridines as well as to phthalans and phthalides. The importance of the aziridine N-substituent in this DoM reaction is stressed as well.
