Palladium-Catalyzed Cross-Coupling Reactions of 4-Tosyl­oxyquinazolines with Indoles: An Efficient Approach to 4-(1H-Indol-1-yl)quinazolines

Palladium-Catalyzed Cross-Coupling Reactions of 4-Tosyl­oxyquinazolines with Indoles: An Efficient Approach to 4-(1H-Indol-1-yl)quinazolines
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钯催化的 4-甲苯磺酰氧基喹唑啉与吲哚的交叉偶联反应：制备 4-(1H-吲哚-1-基)喹唑啉的有效方法

DOI：
10.1055/s-0040-1707356
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发表时间：
2020
期刊：
Synthesis
影响因子：
--
通讯作者：
Peng Yiyuan
Peng Yiyuan
中科院分区：
其他
文献类型：
--
作者：
Ye Xinglin;Huang Jian;Deng Zhihong;Yuan Jianjun;Peng Yiyuan

文献摘要

相似文献

在本文中，描述了我们对喹氮啉核心后期衍生的持续兴趣的探索。在温和的反应条件下，通过钯催化的 4-甲苯磺酰氧基喹唑啉与吲哚衍生物的交叉偶联，以良好至优异的收率获得了多种 4-(1H-吲哚-1-基)喹唑啉。
In this paper, exploration of our continuous interests on late-stage derivation of quinozaline core is described. A wide array of 4-(1H-indol-1-yl)quinazolines were obtained in good to excellent yields through palladium-catalyzed cross-coupling of 4-tosyloxyquinazolines with indole derivatives under mild reaction conditions.