Pharmacokinetics of Propofol and Extrahepatic UGT1A6 Gene Expression in Anhepatic Rats

Pharmacokinetics of Propofol and Extrahepatic UGT1A6 Gene Expression in Anhepatic Rats
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无肝大鼠丙泊酚药代动力学及肝外UGT1A6基因表达

DOI:
10.1159/000236523
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发表时间:
2009-09
期刊:
影响因子:
3.1
通讯作者:
Ma, Daqing
Ma, Daqing
中科院分区:
医学4区
文献类型:
--
作者:
Xia, Peiyuan;Tang, Min;Tao, Guocai;Dai, Qing;Lu, Kaizhi;Gu, Jianteng;Ma, Daqing

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目的:研究认为糖醛酸苷基转移酶1A6 (UGT1A6)代谢酶在肝内或肝外代谢异丙酚。本研究的目的是研究异丙酚的药代动力学和UGT1A6 mRNA的表达
Objective: The metabolic enzyme of UDP-glucuronosyltransferase 1A6 (UGT1A6) has been considered to metabolize propofol intra- or extrahepatically. The aim of the present study was to investigate the pharmacokinetics of propofol and UGT1A6 mRNA expression
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