3-Thio-1,2,4-triazoles, novel somatostatin sst2/sst5 agonists

3-Thio-1,2,4-triazoles, novel somatostatin sst2/sst5 agonists
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DOI:
10.1016/j.bmcl.2005.05.061
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发表时间:
2005-08-01
影响因子:
2.7
通讯作者:
Roubert, P
Roubert, P
中科院分区:
医学4区
文献类型:
--
作者:
Contour-Galcéra, MO;Sidhu, A;Roubert, P

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新的3-硫代1,2,4-三唑通过液相平行合成策略获得,提供有效的非肽类人生长抑素受体亚型2和5激动剂。(c) 2005 Elsevier Ltd版权所有。
Novel 3-thio-1,2,4-triazoles have been obtained via a solution-phase parallel synthesis strategy, affording potent non-peptidic human somatostatin receptor subtypes 2 and 5 agonists. (c) 2005 Elsevier Ltd. All rights reserved.