An efficient and concise synthesis of Indiacen A and Indiacen B
An efficient and concise synthesis of Indiacen A and Indiacen B
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DOI：
10.1016/j.tetlet.2017.03.002
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发表时间：
2017-04-12
影响因子：
1.8
通讯作者：
Maringanti, Thirumala Chary
中科院分区：
文献类型：
--
作者：
Anantoju, Kishore Kumar;Mohd, Baquer Syed;Maringanti, Thirumala Chary
以Horner-Wadsworth-Emmons烯化反应、碳铝化反应、氯化反应和Vilsmeier-Haack加成反应为关键反应，合成了具有抗菌活性的异戊烯基吲哚类化合物Indiacen A及其氯代类似物Indiacen B。(C)2017爱思唯尔有限公司版权所有。
A novel total synthesis of antimicrobial prenyl indoles, Indiacen A and its chloro analogue Indiacen B has been accomplished by using Horner-Wadsworth-Emmons olefination for terminal conjugated enynes, carboalumination, chlorination and Vilsmeier-Haack formylation as the key transformations. (C) 2017 Elsevier Ltd. All rights reserved.