Kinetic analysis of protein kinase C inhibition by staurosporine: evidence that inhibition entails inhibitor binding at a conserved region of the catalytic domain but not competition with substrates.
Kinetic analysis of protein kinase C inhibition by staurosporine: evidence that inhibition entails inhibitor binding at a conserved region of the catalytic domain but not competition with substrates.
复制标题
星形孢菌素对蛋白激酶 C 抑制的动力学分析:证据表明抑制需要抑制剂在催化结构域的保守区域结合,而不是与底物竞争。
作者:
Ward,NE;O'Brian,CA