Kinetic analysis of protein kinase C inhibition by staurosporine: evidence that inhibition entails inhibitor binding at a conserved region of the catalytic domain but not competition with substrates.

Kinetic analysis of protein kinase C inhibition by staurosporine: evidence that inhibition entails inhibitor binding at a conserved region of the catalytic domain but not competition with substrates.
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星形孢菌素对蛋白激酶 C 抑制的动力学分析:证据表明抑制需要抑制剂在催化结构域的保守区域结合,而不是与底物竞争。

DOI:
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发表时间:
1992
影响因子:
3.6
通讯作者:
O'Brian,CA
O'Brian,CA
中科院分区:
医学3区
文献类型:
--
作者:
Ward,NE;O'Brian,CA

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