New aryl/heteroaryl C-N bond cross-coupling reactions via arylboronic acid cupric acetate arylation
New aryl/heteroaryl C-N bond cross-coupling reactions via arylboronic acid cupric acetate arylation
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DOI：
10.1016/s0040-4039(98)00504-8
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发表时间：
1998-05-07
影响因子：
1.8
通讯作者：
Combs, A
中科院分区：
文献类型：
--
作者：
Lam, PYS;Clark, CG;Combs, A
发现了一种新的芳基硼酸/乙酸铜芳基化含N-H杂芳烃的芳基/杂芳基C-N键交叉偶联反应。这种新方法温和，在室温下暴露于空气中进行，并适用于许多杂环芳烃和芳基硼酸，提供了n -芳基杂环芳烃的良好收率。1998爱思唯尔科学有限公司版权所有。
A new aryl/heteroaryl C-N bond cross-coupling reaction via the arylboronic acid/cupric acetate arylation of N-H containing heteroarenes has been discovered. This new methodology is mild, proceeds at room temperature exposed to air, and works for many heteroarenes and arylboronic acids providing good yields of N-arylated heteroarenes. (C) 1998 Elsevier Science Ltd. All rights reserved.