Synthesis of substituted 8-aminoquinolines and phenanthrolines through a Povarov approach
Synthesis of substituted 8-aminoquinolines and phenanthrolines through a Povarov approach
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DOI：
10.1039/c0ob00496k
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发表时间：
2011-01-01
影响因子：
3.2
通讯作者：
Bonnet-Delpona, Daniele
中科院分区：
文献类型：
--
作者：
De, Kavita;Legros, Julien;Bonnet-Delpona, Daniele
The synthesis of 8-aminoquinolines and 1,10-phenanthrolines with substituents in alpha of the nitrogen has been performed through an inverse-demanding aza-Diels-Alder (Povarov reaction) in the fluoroalcohols TFE or HFIP. This path involves simple starting materials: 1,2-phenylenediamines, enol ethers and aldehydes.
