Pd-catalyzed addition of boronic acids to vinylogous imines: a convenient approach to 3-sec-alkyl substituted indoles
Pd-catalyzed addition of boronic acids to vinylogous imines: a convenient approach to 3-sec-alkyl substituted indoles
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DOI：
10.1016/j.tetlet.2012.05.056
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发表时间：
2012-07-25
影响因子：
1.8
通讯作者：
Jiang, Guo-Fang
中科院分区：
文献类型：
--
作者：
Cao, Liang-Liang;Li, Xu-Ni;Jiang, Guo-Fang
通过在温和条件下将芳基硼酸与磺酰吲哚原位生成的插烯亚胺在钯催化下加成，开发了一种制备 3-仲烷基取代吲哚的简便方法。 (C) 2012 Elsevier Ltd. 保留所有权利。
A convenient approach to 3-sec-alkyl substituted indoles was developed via palladium-catalyzed addition of arylboronic acids to vinylogous imines generated in situ from sulfonylindoles under mild conditions. (C) 2012 Elsevier Ltd. All rights reserved.