Synthesis and Utility of Dihydropyridine Boronic Esters.
Synthesis and Utility of Dihydropyridine Boronic Esters.
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DOI：
10.1002/anie.201510027
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发表时间：
2016-02-05
期刊：
影响因子：
--
通讯作者：
Ready JM
中科院分区：
文献类型：
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作者：
Panda S;Coffin A;Nguyen QN;Tantillo DJ;Ready JM
当通过酰化剂活化时，吡啶硼酸酯与有机金属试剂反应以形成二氢吡啶硼酸酯。该中间体允许获得许多有价值的取代吡啶、二氢吡啶和哌啶产物。
When activated by an acylating agent, pyridine boronic esters react with organometallic reagents to form a dihydropyridine boronic ester. This intermediate allows access to a number of valuable substituted pyridine, dihydropyridine and piperidine products.