Synthesis of 9-phenol-substituted xanthenes by cascade O-insertion/1,6-conjugate addition of benzyne with ortho-hydroxyphenyl substituted para-quinone methides
Synthesis of 9-phenol-substituted xanthenes by cascade O-insertion/1,6-conjugate addition of benzyne with ortho-hydroxyphenyl substituted para-quinone methides
复制标题
通过级联 O-插入/苯炔与邻羟基苯基取代的对醌甲基化物的 1,6-共轭加成合成 9-苯酚取代的呫吨
DOI：
10.1016/j.cclet.2018.04.003
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发表时间：
2019-02-01
影响因子：
9.1
通讯作者：
He, Lin
中科院分区：
文献类型：
--
作者：
Li, Zhijuan;Wang, Weihua;He, Lin
本文报道了邻羟基苯基取代的对醌甲基化物与苯偶姻的级联O-插入/1，6共轭加成反应，得到9-苯酚取代的氧杂蒽，产率49%~ 84%。(C)2018中国化学会、中国医学科学院药物研究所。Elsevier B. V.出版，保留所有权利。
The cascade O-insertion/1,6 conjugate addition between benzynes and ortho-hydroxyphenyl substituted para-quinone methides has been reported, affording 9-phenol substituted xanthenes in 49%-84% yields. (C) 2018 Chinese Chemical Society and Institute of Materia Medica, Chinese Academy of Medical Sciences. Published by Elsevier B.V. All rights reserved.