A Novel Indium-Catalyzed Three-Component Reaction: General and Efficient One-Pot Synthesis of Substituted Pyrroles
A Novel Indium-Catalyzed Three-Component Reaction: General and Efficient One-Pot Synthesis of Substituted Pyrroles
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一种新型的铟催化三组分反应：取代吡咯的通用高效一锅法合成
DOI：
10.1055/s-0030-1258525
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发表时间：
2010-09-01
期刊：
影响因子：
2
通讯作者：
Zhan, Zhuang-ping
中科院分区：
文献类型：
--
作者：
Lin, Min;Hao, Lu;Zhan, Zhuang-ping
介绍了一种由炔丙基乙酸酯、烯醇醚和伯胺合成取代吡咯的简便而通用的方法。这种新的转化是在铟的催化下一锅合成的，并获得了各种吡咯衍生物的高产率。
A convenient and general approach towards the synthesis of substituted pyrroles from propargylic acetates, silyl enol ethers, and primary amines was described. This novel transformation was catalyzed by indium trichloride in a one-pot synthesis, and high yields of various pyrrole derivatives were obtained.