Direct synthesis of unprotected 4-aryl phenylalanines via the Suzuki reaction under microwave irradiation.
Direct synthesis of unprotected 4-aryl phenylalanines via the Suzuki reaction under microwave irradiation.
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DOI：
10.1021/ol026587z
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发表时间：
2002-10
期刊：
影响因子：
5.2
通讯作者：
Y. Gong;Wei He
中科院分区：
文献类型：
--
作者：
Y. Gong;Wei He
[公式：在微波辐射下，在5-10分钟内以高产率从4-硼基苯丙氨酸与芳基卤化物的Suzuki偶联制备游离氨基酸形式的4-芳基苯丙氨酸。
[formula: see text] 4-Aryl phenylalanines were prepared as free amino acids from the Suzuki coupling of 4-borono phenylalanine with aryl halides in high yields within 5-10 min under microwave irradiation.