Concise synthesis of oxindole derivatives bearing a 3-trifluoroethyl group: Copper-catalyzed trifluoromethylation of acryloanilides
Concise synthesis of oxindole derivatives bearing a 3-trifluoroethyl group: Copper-catalyzed trifluoromethylation of acryloanilides
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DOI：
10.1016/j.jfluchem.2013.03.009
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发表时间：
2013-08-01
影响因子：
1.9
通讯作者：
Sodeoka, Mikiko
中科院分区：
文献类型：
--
作者：
Egami, Hiromichi;Shimizu, Ryo;Sodeoka, Mikiko
使用 CuI 和 Togni 试剂组合对丙烯酰苯胺衍生物进行碳三氟甲基化，在温和条件下以高产率提供带有 3-三氟乙基的羟吲哚衍生物，且与各种官能团相容。 (c) 2013 Elsevier B.V. 保留所有权利。
Carbotrifluoromethylation of acryloanilide derivatives with the combination of CuI and Togni's reagent affords oxindole derivatives bearing a 3-trifluoroethyl group in high yields under mild conditions that are compatible with various functional groups. (c) 2013 Elsevier B.V. All rights reserved.