An improved method for the palladium-catalyzed amination of aryl iodides
An improved method for the palladium-catalyzed amination of aryl iodides
复制标题
DOI：
10.1021/jo0008486
复制
发表时间：
2001-04-20
影响因子：
3.6
通讯作者：
Buchwald, SL
中科院分区：
文献类型：
--
作者：
Ali, MH;Buchwald, SL
在钯、合适的配体和Naot-Bu的存在下，芳基碘与胺偶联，以高产率得到相应的芳胺。当Cs2CO3被取代为碱时，功能化的芳基碘可以很好地得到相应的芳胺。
Aryl iodides are coupled with amines to give the corresponding arylamines in high yield in the presence of palladium, a suitable ligand, and NaOt-Bu. Functionalized aryl iodides give good yields of the corresponding arylamines when Cs2CO3 is substituted as the base.