Regioselective Synthesis of Diltiazem Analogue Pyrazolo[4,3-c][1,5]benzothiazepines and Antifungal Activity
Regioselective Synthesis of Diltiazem Analogue Pyrazolo[4,3-c][1,5]benzothiazepines and Antifungal Activity
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DOI：
10.1080/10426501003713064
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发表时间：
2010-11
期刊：
影响因子：
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通讯作者：
A. Dandia;Ruby Singh;Dharmendra Singh;Ashok K. Laxkar;Asha Sivpuri
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文献类型：
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作者：
A. Dandia;Ruby Singh;Dharmendra Singh;Ashok K. Laxkar;Asha Sivpuri
A dry media procedure has been developed for the synthesis of a series of new class of pyrazolo [4,3-c][1,5]benzothiazepines 6 under microwave irradiation using montmorillonite K10 as solid support. The catalyst can be recovered and reused. Thus, the procedure provides a simple and green synthetic methodology under environmentally friendly conditions. Antifungal screening of synthesized compounds has shown promising activity. Supplemental materials are available for this article. Go to the publisher's online edition of Phosphorus, Sulfur, and Silicon and the Related Elements to view the free supplemental file.
