K-252A, A POTENT INHIBITOR OF PROTEIN-KINASE-C FROM MICROBIAL ORIGIN

K-252A, A POTENT INHIBITOR OF PROTEIN-KINASE-C FROM MICROBIAL ORIGIN
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DOI:
10.7164/antibiotics.39.1059
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发表时间:
1986-08-01
影响因子:
3.3
通讯作者:
MATSUDA, Y
MATSUDA, Y
中科院分区:
医学4区
文献类型:
--
作者:
KASE, H;IWAHASHI, K;MATSUDA, Y

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K-252a,从诺卡氏菌培养液中分离出来的代谢物。 K-252a被发现对蛋白激酶C表现出极强的抑制活性。IC50值为32.9 nM。
K-252a, a metabolite isolated from the culture broth of Nocardiopsis sp. K-252a, was found to exhibit an extremely potent inhibitory activity on protein kinase C. The IC50 value was 32.9 nM.