Regioselective syntheses of fully-substituted 1,2,3-triazoles: the CuAAC/C-H bond functionalization nexus
Regioselective syntheses of fully-substituted 1,2,3-triazoles: the CuAAC/C-H bond functionalization nexus
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DOI：
10.1039/c0ob00212g
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发表时间：
2010-01-01
影响因子：
3.2
通讯作者：
Potukuchi, Harish Kumar
中科院分区：
文献类型：
--
作者：
Ackermann, Lutz;Potukuchi, Harish Kumar
1，4，5-三取代-1，2，3-三唑的区域选择性合成是通过三种不同的策略完成的，依赖于(I)化学计量形成的5-铜-1，2，3-三唑的截取，(Ii)化学计量官能化炔烃的使用或(Iii)催化C-H键官能化。这篇前瞻性文章总结了截至2010年6月在这一研究领域取得的进展。
Regioselective syntheses of 1,4,5-trisubstituted 1,2,3- triazoles were accomplished by three different strategies, relying on (i) the interception of stoichiometrically formed 5-cuprated-1,2,3-triazoles, (ii) the use of stoichiometrically functionalized alkynes or (iii) catalytic C-H bond functionalizations. This perspective article summarizes progress in this research area until June 2010.