Aromatic amines as nucleophiles in the Bargellini reaction
Aromatic amines as nucleophiles in the Bargellini reaction
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DOI：
10.1016/j.tetlet.2009.03.044
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发表时间：
2009-05-27
影响因子：
1.8
通讯作者：
Hurst, Jenny
中科院分区：
文献类型：
--
作者：
Butcher, Ken J.;Hurst, Jenny
芳族胺可用于Bargellini反应以产生有用的中间体。快速，实用的功能化，特权结构的访问可能有显着的效用在药物样分子的合成。卡芬太尼类似物的改进合成说明了这一点。(C)2009爱思唯尔有限公司保留所有权利。
Aromatic amines can be employed in the Bargellini reaction to generate useful intermediates. Rapid, practical access to functionalised, privileged structures may have significant utility in the synthesis of drug-like molecules. An improved synthesis of carfentanil analogues illustrates this point. (C) 2009 Elsevier Ltd. All rights reserved.