Fragment-based screening sees the light

Fragment-based screening sees the light
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基于片段的筛选迎来曙光

DOI:
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发表时间:
2020
期刊:
Nature reviews. Drug discovery
影响因子:
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通讯作者:
Asher Mullard
Asher Mullard
中科院分区:
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文献类型:
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作者:
Asher Mullard

文献摘要

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基于片段的筛选方法正在激增,这是对新目标空间和靶向降解物的兴趣所推动的。基于片段的筛选方法正在激增,这是对新目标空间和靶向降解物的兴趣所推动的。
Fragment-based screening methodologies are proliferating, fuelled by interest in novel target space and targeted degraders. Fragment-based screening methodologies are proliferating, fuelled by interest in novel target space and targeted degraders.