Development of an oral satraplatin pharmaceutical formulation by encapsulation with cyclodextrin

Development of an oral satraplatin pharmaceutical formulation by encapsulation with cyclodextrin
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通过环糊精封装开发口服沙铂药物制剂

DOI:
10.1039/c5ra27182g
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发表时间:
2016-02
期刊:
影响因子:
3.9
通讯作者:
Jun Lin
Jun Lin
中科院分区:
化学3区
文献类型:
--
作者:
Ke Li;Kun-Ming Jiang;Yi Jin;Jun Lin

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制备了一种新型的水溶性口服沙铂/β-环糊精包合物,并对其进行了表征。通过分子动力学模拟研究了其包结机理。通过环糊精包封实现
A novel water-soluble oral satraplatin/β-cyclodextrin inclusion complex was prepared and characterized with a variety of techniques. Molecular dynamics simulations were performed to clarify its inclusion mechanism. Enabled by encapsulation with cyclodextr
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