An efficient and highly regioselective fluorination of aziridines using BF3•OEt2 as fluorine source
An efficient and highly regioselective fluorination of aziridines using BF3•OEt2 as fluorine source
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DOI：
10.1055/s-2004-831319
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发表时间：
2004-10-01
期刊：
影响因子：
2
通讯作者：
Hou, XL
中科院分区：
文献类型：
--
作者：
Ding, CH;Dai, LX;Hou, XL
以氮杂环丙烷和三氟化硼为原料，高区域选择性、高收率地合成了β-氟代胺。（BF 3 OEt 2）-O-的所有三个氟原子。当它与氮丙啶反应时被掺入到产物中。
beta-Fluoro amines were prepared from the reaction of aziridines and boron trifluoride in high regioselectivity and in high yield. All three fluorine atoms of (BF3OEt2)-O-. were incorporated into the products when it reacted with aziridines.