An efficient one-pot procedure for the synthesis of 1,5-benzothiazepinones catalyzed by tetrabutylammonium fluoride (TBAF)
An efficient one-pot procedure for the synthesis of 1,5-benzothiazepinones catalyzed by tetrabutylammonium fluoride (TBAF)
复制标题
四丁基氟化铵 (TBAF) 催化合成 1,5-苯并硫氮杂酮的高效一锅法
DOI：
10.1016/j.tetlet.2016.07.012
复制
发表时间：
2016-08-17
影响因子：
1.8
通讯作者：
Chu, Yong
中科院分区：
文献类型：
--
作者：
Zhang, Peng;Ye, Deyong;Chu, Yong
以四丁基氟化铵（TBAF）为催化剂，开发了一种实用高效、产率高的1,5-苯并噻吩类酮衍生物的制备方法。本研究不仅扩展了以往对底物的研究范围，而且对这类药物支架的化学性质有了更多的了解。(C) 2016 Elsevier Ltd.版权所有。
A practical and efficient method for the preparation of 1,5-benzothiazepinone derivatives in good yields has been developed using tetrabutylammonium fluoride (TBAF) as a catalyst. This study not only expands the previous work on the substrate scope and also provides more understanding of the chemistry of such drug scaffolds. (C) 2016 Elsevier Ltd. All rights reserved.