Design, synthesis and structure-activity relationships of (indo-3-yl) heterocyclic derivatives as agonists of the CB1 receptor. Discovery of a clinical candidate.
Design, synthesis and structure-activity relationships of (indo-3-yl) heterocyclic derivatives as agonists of the CB1 receptor. Discovery of a clinical candidate.
复制标题
作为 CB1 受体激动剂的 (indo-3-yl) 杂环衍生物的设计、合成和构效关系。
DOI:
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发表时间:
2011
影响因子:
2.7
通讯作者:
J. I. Udo de Haes
中科院分区:
文献类型:
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作者:
P. Ratcliffe;Julia M. Adam;James Baker;R. Bursi;Robert A. Campbell;J. Clark;J. Cottney;M. Deehan;Anna;Daniel Ecker;Darren Edwards;O. Epemolu;Louise S. Evans;Ruth Fields;S. Francis;Paul J. Harradine;Fiona Jeremiah;T. Kiyoi;D. Mcarthur;Angus J. Morrison;P. Passier;J. Pick;P. G. Schnabel;J. Schulz;H. Steinbrede;G. Walker;P. Westwood;G. Wishart;J. I. Udo de Haes