Efficient Synthesis of 2‐Fluoromethylated Quinolines via Copper‐Catalyzed Alkynylation and Cyclization of Fluorinated Imidoyl Iodides
Efficient Synthesis of 2‐Fluoromethylated Quinolines via Copper‐Catalyzed Alkynylation and Cyclization of Fluorinated Imidoyl Iodides
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DOI：
10.1002/adsc.201000180
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发表时间：
2010-07
影响因子：
5.4
通讯作者：
Shan Li;Yafen Yuan;Jiangtao Zhu;Haibo Xie;Zixian Chen;Yong-ming Wu
中科院分区：
文献类型：
--
作者：
Shan Li;Yafen Yuan;Jiangtao Zhu;Haibo Xie;Zixian Chen;Yong-ming Wu
2-氟甲基喹啉是由N-芳基-氟化亚胺基碘与末端炔在单独的碘化铜(CuI)催化下以较高的产率合成的。
2-Fluoromethylated quinolines were synthesized through the reaction of N-aryl-fluorinated imidoyl iodides with terminal alkynes in good yields by the catalysis of copper(I) iodide (CuI) alone.