The discovery of novel histone lysine methyltransferase G9a inhibitors (part 1): molecular design based on a series of substituted 2,4-diamino-7- aminoalkoxyquinazoline by molecular-docking-guided 3D quantitative structure-activity relatio
The discovery of novel histone lysine methyltransferase G9a inhibitors (part 1): molecular design based on a series of substituted 2,4-diamino-7- aminoalkoxyquinazoline by molecular-docking-guided 3D quantitative structure-activity relatio
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新型组蛋白赖氨酸甲基转移酶 G9a 抑制剂的发现(第 1 部分):基于一系列取代的 2,4-二氨基-7-氨基烷氧基喹唑啉,通过分子对接引导的 3D 定量构效关系进行分子设计
作者:
Feng, Taotao;Wang, Hai;Zhang, Xiaojin;Sun, Haopeng;You, Qidong