Aromatic Enamide/Ene Metathesis toward Substituted Indoles and Its Application to the Synthesis of Indomethacins
Aromatic Enamide/Ene Metathesis toward Substituted Indoles and Its Application to the Synthesis of Indomethacins
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DOI：
10.1002/ejoc.200900520
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发表时间：
2009-09-01
影响因子：
2.8
通讯作者：
Arisawa, Mitsuhiro
中科院分区：
文献类型：
--
作者：
Kasaya, Yayoi;Hoshi, Kosuke;Arisawa, Mitsuhiro
介绍了烯酰胺/烯复分解反应的空间和电子效应，以烯酰胺/烯复分解反应为关键反应制备2-取代吲哚和3-取代吲哚的新方法，以及在吲哚美辛合成中的应用。((C)Wiley-VCH Verlag GmbH & Co. KGaA，69451魏因海姆，德国，2009）
A steric and electronic effect on enamide/ene metathesis, a novel preparation of 2-substituted indoles and 3-substituted indoles using enamide-ene metathesis as a key reaction, and its application to the synthesis of indomethacin are described. ((C) Wiley-VCH Verlag GmbH & Co. KGaA, 69451 Weinheim, Germany, 2009)