Preparation and Utility of 5-β-D-Ribofuranosyl-1H-tetrazole as a Key Synthon for C-Nucleoside Synthesis
Preparation and Utility of 5-β-D-Ribofuranosyl-1H-tetrazole as a Key Synthon for C-Nucleoside Synthesis
复制标题
5-β-D-呋喃核糖基-1H-四唑的制备及其作为 C-核苷合成关键合成子的应用
DOI：
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发表时间：
1994
期刊：
影响因子：
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通讯作者：
L. Townsend
中科院分区：
文献类型：
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作者：
J. Kobe;M. Prhavc;M. Hohnjec;L. Townsend
本文报道了5-β-D-呋喃核糖基-1H-四唑(2)和呋喃核苷(9)衍生物的合成。为了确定该合成子的稳定性，进一步用于偶极环加成反应，研究了2的环变换。
Abstract A synthesis of 5-β-D-ribofuranosyl-1H-tetrazole (2) and 5-β-D-ribo-furanosyl-1,3,4-oxadiazole-2(3H)-one (9) derivatives is described. Ring transformations of 2 have been investigated in an effort to establish the stability of this synthon for further use in dipolar cycloaddition reactions.