Discovery of (E)-N-(4-((4-methylpiperazin-1-yl)methyl)-3-(trifluoromethyl)phenyl)-3-((3-(2-(py ridin-2-yl)vinyl)-1H-indazol-6-yl)thio)propanamide (CHMFL-ABL-121) as a highly potent ABL kinase inhibitor capable of overcoming a variety of ABL mutants includ

Discovery of (E)-N-(4-((4-methylpiperazin-1-yl)methyl)-3-(trifluoromethyl)phenyl)-3-((3-(2-(py ridin-2-yl)vinyl)-1H-indazol-6-yl)thio)propanamide (CHMFL-ABL-121) as a highly potent ABL kinase inhibitor capable of overcoming a variety of ABL mutants includ
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(E)-N-(4-((4-甲基哌嗪-1-基)甲基)-3-(三氟甲基)苯基)-3-((3-(2-(吡啶-2-基)乙烯基)的发现

DOI:
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发表时间:
2018
期刊:
Eur J Med Chem
影响因子:
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通讯作者:
Wenchao Wang
Wenchao Wang
中科院分区:
其他
文献类型:
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作者:
Wenchao Wang

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