Indole synthesis through transition metal-catalyzed C-H activation
Indole synthesis through transition metal-catalyzed C-H activation
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DOI：
10.1016/j.tetlet.2014.11.114
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发表时间：
2015-01-08
影响因子：
1.8
通讯作者：
Yu, Zhengkun
中科院分区：
文献类型：
--
作者：
Guo, Tenglong;Huang, Fei;Yu, Zhengkun
吲哚的合成是氮杂环化学中最重要的任务之一。已经开发了多种合成方法来建立吲哚主链，但人们强烈希望获得吲哚衍生物的简明和直接的途径。本文综述了近五年来过渡金属催化C-H活化法合成吲哚的主要进展。对这些合成协议的可能应用进行了简要的讨论。(C)2014爱思唯尔有限公司。保留所有权利。
Indole synthesis is among one of the most important tasks in N-heterocyclic chemistry. Versatile synthetic methods have been developed for the establishment of an indole backbone, but concise and straightforward routes to access indole derivatives have been strongly desired. This digest paper summarizes the major advances in catalytic synthesis of indoles through transition-metal-catalyzed C-H activation during the last five years. Brief discussions are given for possible applications of these synthetic protocols. (C) 2014 Elsevier Ltd. All rights reserved.