Iodine-catalyzed oxidative annulation of 3-cyanoacetylindoles with benzylamines: facile access to 5-(3-indolyl)oxazoles
Iodine-catalyzed oxidative annulation of 3-cyanoacetylindoles with benzylamines: facile access to 5-(3-indolyl)oxazoles
复制标题
碘催化 3-氰基乙酰吲哚与苄胺的氧化环化：轻松获得 5-(3-吲哚基)恶唑
DOI：
10.1039/c8ob00833g
复制
发表时间：
2018-05-21
影响因子：
3.2
通讯作者：
Liu, Peijun
中科院分区：
文献类型：
--
作者：
Liu, Xiaozu;Zhou, Yuxiang;Liu, Peijun
已经开发出一种碘催化的 3-氰基乙酰吲哚与苄胺的氧化成环反应。该反应能够在温和的条件下方便地合成各种具有广泛官能团兼容性的5-(3-吲哚基)恶唑。
An iodine-catalyzed oxidative annulation of 3-cyanoacetylindoles with benzylamines has been developed. This reaction enables the convenient synthesis of a variety of 5-(3-indolyl)oxazoles under mild conditions with broad functional group compatibility.