Cobalt (II)-catalyzed direct C3-selective C–H acyloxylation of indoles with tert-butyl peresters
Cobalt (II)-catalyzed direct C3-selective C–H acyloxylation of indoles with tert-butyl peresters
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DOI：
10.1080/00397911.2018.1524493
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发表时间：
2018-11
影响因子：
2.1
通讯作者：
Yuxiang Zhou;Guojun Chen;Chenglong Li;Xiaozu Liu;Peijun Liu
中科院分区：
文献类型：
--
作者：
Yuxiang Zhou;Guojun Chen;Chenglong Li;Xiaozu Liu;Peijun Liu
Abstract A Co(II)-catalyzed direct C3-selective C–H acyloxylation of indoles has been realized with tert-butyl peresters serving as both an acyloxy source and an oxidant. This reaction features highly C3 regioselectivity and good functional group tolerance, which provides a convenient and versatile approach to the construction of valuable 3-acyloxyindoles in moderate to excellent yields. Graphical Abstract
