Synthesis and Biological Evaluation of Some Pyrazole Derivatives, Containing (Thio) Semicarbazide, as Dual Anti-Inflammatory Antimicrobial Agents

Synthesis and Biological Evaluation of Some Pyrazole Derivatives, Containing (Thio) Semicarbazide, as Dual Anti-Inflammatory Antimicrobial Agents
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某些含(硫代)氨基脲的吡唑衍生物作为双重抗炎抗菌剂的合成及生物学评价

DOI:
10.2174/1570180816666190325163117
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发表时间:
2019-08
影响因子:
1
通讯作者:
Deng Xianqing
Deng Xianqing
中科院分区:
医学4区
文献类型:
--
作者:
Liang Zhaochang;Huang Yuping;Wang Shiben;Deng Xianqing

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设计并合成了几个系列的含(硫代)氨基脲的吡唑衍生物(4a-4 h,5a-5l,6a-6 f,7a-7 c),并进行了抗炎和抑菌双重活性的筛选。产物经1H NMR、13 C NMR和HRMS表征。在v
Several series of pyrazole derivatives containing (thio) semicarbazide (4a-4h, 5a-5l, 6a-6f, 7a-7c) were designed and synthesized to screen dual inflammatory and antimicrobial activities. The products were characterized by1H NMR, 13C NMR and HRMS. In v
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