Discovery of an SphK1 inhibitor: A hybrid approach involving a receptor–ligand-complex-based pharmacophore and docking-based virtual screening
Discovery of an SphK1 inhibitor: A hybrid approach involving a receptor–ligand-complex-based pharmacophore and docking-based virtual screening
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SphK1 抑制剂的发现:涉及基于受体配体复合物的药效基团和基于对接的虚拟筛选的混合方法
DOI:
10.1177/17475198221089222
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发表时间:
2022-03
影响因子:
1.4
通讯作者:
Bo Liu
中科院分区:
文献类型:
--
作者:
Ti;i Ding;HaiJiao Chen;Yan Li;Ying Li;Ying Zhi;Zhiqiang Qu;Qiang Sun;Qingqiang Yao;Bo Liu
Sphingosine kinase is a lipid kinase that catalyzes the phosphorylation of sphingosine to sphingosine-1-phosphate. Sphingosine-1-phosphate is a bioactive lipid that regulates biological processes. The overexpression of sphingosine kinases is related to a
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