Discovery of an SphK1 inhibitor: A hybrid approach involving a receptor–ligand-complex-based pharmacophore and docking-based virtual screening

Discovery of an SphK1 inhibitor: A hybrid approach involving a receptor–ligand-complex-based pharmacophore and docking-based virtual screening
复制标题

SphK1 抑制剂的发现:涉及基于受体配体复合物的药效基团和基于对接的虚拟筛选的混合方法

DOI:
10.1177/17475198221089222
复制
发表时间:
2022-03
影响因子:
1.4
通讯作者:
Bo Liu
Bo Liu
中科院分区:
化学4区
文献类型:
--
作者:
Ti;i Ding;HaiJiao Chen;Yan Li;Ying Li;Ying Zhi;Zhiqiang Qu;Qiang Sun;Qingqiang Yao;Bo Liu

文献摘要

参考文献

相似文献

鞘氨醇激酶是催化鞘氨醇磷酸化为鞘氨醇-1-磷酸的脂质激酶。鞘氨醇-1-磷酸是一种调节生物过程的生物活性脂质。鞘氨醇激酶的过度表达与
Sphingosine kinase is a lipid kinase that catalyzes the phosphorylation of sphingosine to sphingosine-1-phosphate. Sphingosine-1-phosphate is a bioactive lipid that regulates biological processes. The overexpression of sphingosine kinases is related to a
DOI: 10.1016/j.molstruc.2020.127900
发表时间: 2020-05
影响因子: 3.8
作者:
Jinmiao Zhang;Maoyu Zhang;Jinying Yu;Yanguo Shang;Kaixuan Jiang;Y. Jia;Jin-Xing Wang;Kan Yang-Ka
通讯作者: Jinmiao Zhang;Maoyu Zhang;Jinying Yu;Yanguo Shang;Kaixuan Jiang;Y. Jia;Jin-Xing Wang;Kan Yang-Ka
DOI: 10.1016/j.bmcl.2019.126712
发表时间: 2019-10
影响因子: 2.7
作者:
Feng Li;Qinlong Xu;Qihua Zhu;Zhaoxing Chu;Gaofeng Lin;Jiajia Mo;Yan Zhao;Jiaming Li;Guangwei He;Yungen Xu
通讯作者: Feng Li;Qinlong Xu;Qihua Zhu;Zhaoxing Chu;Gaofeng Lin;Jiajia Mo;Yan Zhao;Jiaming Li;Guangwei He;Yungen Xu
DOI: 10.1016/j.bmcl.2011.08.003
发表时间: 2011-10
影响因子: 2.7
作者:
Iljung Lee;Jehoon Yang;J. H. Lee;Y. Choe
通讯作者: Iljung Lee;Jehoon Yang;J. H. Lee;Y. Choe
DOI: 10.1021/ml5004074
发表时间: 2014-12-01
影响因子: 4.2
作者:
Wang, Jing;Knapp, Stefan;Elkins, Jonathan M.
通讯作者: Elkins, Jonathan M.
DOI: 10.1016/j.tcb.2011.09.003
发表时间: 2012-01
影响因子: 19
作者:
Maceyka, Michael;Harikumar, Kuzhuvelil B.;Milstien, Sheldon;Spiegel, Sarah
通讯作者: Spiegel, Sarah