A new strategy for hit generation: Novel in cellulo active inhibitors of CYP121A1 from Mycobacterium tuberculosis via a combined X-ray crystallographic and phenotypic screening approach (XP screen)
A new strategy for hit generation: Novel in cellulo active inhibitors of CYP121A1 from Mycobacterium tuberculosis via a combined X-ray crystallographic and phenotypic screening approach (XP screen)
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命中生成的新策略:通过结合 X 射线晶体学和表型筛选方法(XP 筛选)从结核分枝杆菌中获得新型 CYP121A1 纤维素活性抑制剂
DOI:
10.25418/crick.20383548
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发表时间:
2022
期刊:
影响因子:
--
通讯作者:
Frederickson M
中科院分区:
文献类型:
--
作者:
Frederickson M
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影响因子:
15
作者:
Knapp DM;Gillis EP;Burke MD
通讯作者:
Burke MD
影响因子:
4.1
作者:
C. Leadbeater;L. McIver;D. Campopiano;S. Webster;R. Baxter;S. Kelly;N. C. Price;D. A. Lysek;M. Noble;S. Chapman;A. Munro
通讯作者:
A. Munro
影响因子:
64.8
作者:
T. Ely
通讯作者:
T. Ely
影响因子:
3.4
作者:
Kavanagh, Madeline E.;Gray, Janine L.;Gilbert, Sophie H.;Coyne, Anthony G.;McLean, Kirsty J.;Davis, Holly J.;Munro, Andrew W.;Abell, Chris
通讯作者:
Abell, Chris
影响因子:
4.1
作者:
Leadbeater, C;McIver, L;Munro, AW
通讯作者:
Munro, AW