Modifying ICCA with Trp-Phe-Phe to Enhance in vivo Activity and Form Nano-Medicine

Modifying ICCA with Trp-Phe-Phe to Enhance in vivo Activity and Form Nano-Medicine
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Trp-Phe-Phe修饰ICCA增强体内活性形成纳米药物

DOI:
10.2147/ijn.s229856
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发表时间:
2020-01
影响因子:
8
通讯作者:
Peng Shiqi
Peng Shiqi
中科院分区:
医学2区
文献类型:
--
作者:
Zhang Xiaoyi;Zhang Yixin;Wang Yaonan;Wu Jianhui;Chen Haiyan;Zhao Ming;Peng Shiqi

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1-(4-异丙基苯基)-β-咔啉-3-羧酸(ICCA)经Trp-Phe-Phe修饰,得到1-(4-异丙基苯基)-β-咔啉-3-羰基-Trp-Phe-Phe(ICCA-WFF)。目的制备ICCA-WFF,以提高ICCA-WFF的体内药效。
Background 1-(4-isopropylphenyl)-β-carboline-3-carboxylic acid (ICCA) was modified by Trp-Phe-Phe to form 1-(4-isopropylphenyl)-β-carboline-3-carbonyl-Trp-Phe-Phe (ICCA-WFF). Purpose The object of preparing ICCA-WFF was to enhance the in vivo efficacy of
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