Co‐administration of nuciferine reduces the concentration of metformin in liver via differential inhibition of hepatic drug transporter OCT1 and MATE1

Co‐administration of nuciferine reduces the concentration of metformin in liver via differential inhibition of hepatic drug transporter OCT1 and MATE1
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荷叶碱的联合给药通过对肝脏药物转运蛋白 OCT1 和 MATE1 的差异抑制来降低肝脏中二甲双胍的浓度

DOI:
10.1002/bdd.2158
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发表时间:
2018-10
期刊:
Biopharm Drug Dispos
影响因子:
--
通讯作者:
Huidi Jiang
Huidi Jiang
中科院分区:
其他
文献类型:
--
作者:
Liping Li;Hongmei Lei;Wei Wang;Weijuan Du;Jingqun Yuan;Meijuan Tu;Hui Zhou;Su Zeng;Huidi Jiang

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荷叶碱(NF)是荷花中的主要有效成分之一。叶提取物是治疗肥胖相关疾病的有前途的候选药物,而二甲双胍是 2 型糖尿病的一线治疗药物
Nuciferine (NF), one of the main and effective components in Nelumbo nucifera Gaertn. leaf extracts, is a promising drug candidate for the treatment of obesity‐related diseases, while metformin is a first line therapeutic drug for type 2 diabetes mellitus
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