Pharmacokinetics and brain penetration of LF-3-88, (2-[5-[5-(2(S)-azetidinylmethoxyl)-3-pyridyl]-3-isoxazolyl]ethanol), a selective α4β2-nAChR partial agonist and promising antidepressant.
Pharmacokinetics and brain penetration of LF-3-88, (2-[5-[5-(2(S)-azetidinylmethoxyl)-3-pyridyl]-3-isoxazolyl]ethanol), a selective α4β2-nAChR partial agonist and promising antidepressant.
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LF-3-88(2-[5-[5-(2(S)-azetidinylmethoxyl)-3-pyridyl]-3-isoxazolyl]ethanol)的药代动力学和脑渗透性,选择性α4β2-nAChR部分激动剂
DOI:
10.1016/j.jchromb.2012.11.011
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发表时间:
2013
期刊:
影响因子:
--
通讯作者:
vanBreemen,RichardB
中科院分区:
文献类型:
--
作者:
Yuan,Yang;Yu,Li-Fang;Qiu,Xi;Kozikowski,AlanP;vanBreemen,RichardB
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影响因子:
7.3
作者:
Liu, Jianhua;Yu, Li-Fang;Eaton, J. Brek;Caldarone, Barbara;Cavino, Katie;Ruiz, Christina;Terry, Matthew;Fedolak, Allison;Wang, Daguang;Ghavami, Afshin;Lowe, David A.;Brunner, Dani;Lukas, Ronald J.;Kozikowski, Alan P.
通讯作者:
Kozikowski, Alan P.
影响因子:
4.7
作者:
Mineur, Yann S.;Somenzi, Oli;Picciotto, Marina R.
通讯作者:
Picciotto, Marina R.
影响因子:
56.9
作者:
MCGEHEE, DS;HEATH, MJS;ROLE, LW
通讯作者:
ROLE, LW
影响因子:
4.1
作者:
Dunbar, Geoffrey C.;Inglis, Fraser;Wamsley, James
通讯作者:
Wamsley, James
影响因子:
13.8
作者:
Mineur YS;Picciotto MR
通讯作者:
Picciotto MR