Pharmacological characterization of a novel metal-based proteasome inhibitor Na-AuPT for cancer treatment

Pharmacological characterization of a novel metal-based proteasome inhibitor Na-AuPT for cancer treatment
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新型金属蛋白酶体抑制剂 Na-AuPT 用于癌症治疗的药理学特征

DOI:
10.1038/s41401-021-00816-z
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发表时间:
2021-12
期刊:
Acta Pharmacologica Sinica 
影响因子:
--
通讯作者:
Jin-bao Liu
Jin-bao Liu
中科院分区:
其他
文献类型:
--
作者:
Da-cai Xu;Li Yang;Pei-quan Zhang;Ding Yan;Qian Xue;Qing-tian Huang;Xiao-fen Li;Ya-li Hao;Dao-lin Tang;Q. Ping Dou;Xin Chen;Jin-bao Liu

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The ubiquitin-proteasome system (UPS) is essential for maintaining cell homeostasis by orchestrating the protein degradation, but is impaired in various diseases, including cancers. Several proteasome inhibitors, such as bortezomib, are currently used in
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