Binding mode of inhibitors and Cryptosporidium parvum IMP dehydrogenase: A combined ligand- and receptor-based study

Binding mode of inhibitors and Cryptosporidium parvum IMP dehydrogenase: A combined ligand- and receptor-based study
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抑制剂与小隐孢子虫 IMP 脱氢酶的结合模式:基于配体和受体的联合研究

DOI:
10.1080/1062936x.2015.1043341
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发表时间:
2015-05
影响因子:
3
通讯作者:
Cheng Maosheng
Cheng Maosheng
中科院分区:
环境科学与生态学3区
文献类型:
--
作者:
Li Ruijuan;Wang Yali;Wang Qinghe;Huang Wanxu;Wang Jian;Cheng Maosheng

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A combined ligand- and target-based approach was used to analyse the interaction models of Cryptosporidium parvum inosine 5’-monophosphate dehydrogenase (CpIMPDH) with selective inhibitors. First, a ligand-based pharmacophore model was generated from 20 N
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