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TESTING OF ANTIPROGESTATIONAL/POSTCOITAL AGENTS

TESTING OF ANTIPROGESTATIONAL/POSTCOITAL AGENTS
抗孕/性交后药物的测试
批准号:
2315721
负责人:
C EDGAR COOK
金额:
$62.55万
依托单位:
依托单位国家:
美国
项目类别:
财政年份:
1995
资助国家:
美国
项目状态:
已结题
起止时间:
1995-09-01 至 1998-08-31

项目摘要

项目成果

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中文摘要
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英文摘要
The proposed research is a comprehensive, 36-month, synthetic and biological testing program aimed at the development of novel antiprogestational agents that will interfere with progesterone receptor utilization, and that are orally tenfold more potent that mifepristone and have minimal hormonal and antagonistic activity other than antiprogestational. The proposed research may lead to the development of new derivatives of mifepristone that show significantly improved oral antiprogestational potency with less or without antiglucocorticoid activity, and have better pharmacokinetic and solubility characteristics, thus providing a postcoital emergency therapy as well as a new, highly effective, and safe contraceptive agent.
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会议论文
QUANTITATIVE ANALYSIS OF A METHOD DEVELOPMENT FOR CANN
  • 批准号:
    6012819
  • 项目类别:
  • 资助金额:
    $0.0万
  • 财政年份:
    1998
  • 负责人:
    C EDGAR COOK
  • 依托单位:
QUANTITATIVE ANALYSIS OF A METHOD DEVELOPMENT FOR CANN
  • 批准号:
    6031428
  • 项目类别:
  • 资助金额:
    $22.0万
  • 财政年份:
    1998
  • 负责人:
    C EDGAR COOK
  • 依托单位:
QUANTITATIVE ANALYSIS OF A METHOD DEVELOPMENT FOR CANN
  • 批准号:
    2767704
  • 项目类别:
  • 资助金额:
    $22.0万
  • 财政年份:
    1998
  • 负责人:
    C EDGAR COOK
  • 依托单位:
QUANTITATIVE ANALYSIS OF A METHOD DEVELOPMENT FOR CANN
  • 批准号:
    6261437
  • 项目类别:
  • 资助金额:
    $22.0万
  • 财政年份:
    1998
  • 负责人:
    C EDGAR COOK
  • 依托单位:
海外基金