NOVEL ANTIHYPERTENSIVES: RATIONAL DESIGN AND EVALUATION
NOVEL ANTIHYPERTENSIVES: RATIONAL DESIGN AND EVALUATION
批准号:
2216234
负责人:
SHELDON W MAY
金额:
$24.68万
依托单位国家:
美国
项目类别:
财政年份:
1982
资助国家:
美国
项目状态:
已结题
起止时间:
1982-01-01 至 1996-06-30
期刊论文(19)
专著(0)
科研奖励(0)
会议论文
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Demonstration of the antihypertensive activity of phenyl-2-aminoethyl selenide.
证明苯基-2-氨乙基硒化物的抗高血压活性。
DOI:
--
发表时间:
1988
期刊:
The Journal of pharmacology and experimental therapeutics
影响因子:
--
作者:
[Pollock,SH, Herman,HH, Fowler,LC, Edwards,AS, Evans,CO, May,SW]
通讯作者:
May,SW
Interaction of non-conjugated olefinic substrate analogues with dopamine beta-monooxygenase: catalysis and mechanism-based inhibition.
非共轭烯属底物类似物与多巴胺β-单加氧酶的相互作用:催化和基于机制的抑制。
DOI:
10.1042/bj3060077
发表时间:
1995
期刊:
The Biochemical journal
影响因子:
--
作者:
[Sirimanne,SR, May,SW]
通讯作者:
May,SW
Activation of an adrenergic pro-drug through sequential stereoselective action of tandem target enzymes.
通过串联靶酶的连续立体选择性作用激活肾上腺素能前药。
DOI:
10.1016/0006-291x(92)91521-q
发表时间:
1992
期刊:
Biochemical and biophysical research communications
影响因子:
3.1
作者:
[Debnath,J, Husain,PA, May,SW]
通讯作者:
May,SW
Novel antihypertensives targeted at dopamine beta-monooxygenase: turnover-dependent cofactor depletion by phenyl aminoethyl selenide.
针对多巴胺β-单加氧酶的新型抗高血压药:苯氨乙基硒化物导致周转依赖性辅因子消耗。
DOI:
10.1021/jm00401a003
发表时间:
1988
期刊:
Journal of medicinal chemistry
影响因子:
7.3
作者:
[May,SW, Wimalasena,K, Herman,HH, Fowler,LC, Ciccarello,MC, Pollock,SH]
通讯作者:
Pollock,SH
Effects of dopamine beta-monooxygenase substrate analogs on ascorbate levels and norepinephrine synthesis in adrenal chromaffin granule ghosts.
多巴胺β-单加氧酶底物类似物对肾上腺嗜铬颗粒鬼中抗坏血酸水平和去甲肾上腺素合成的影响。
DOI:
--
发表时间:
1989
期刊:
The Journal of biological chemistry
影响因子:
--
作者:
[Wimalasena,K, Herman,HH, May,SW]
通讯作者:
May,SW
共 17 条
NEUROPEPTIDES--APPROACH TO AMIDATION EFFECTORS
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批准号:2022242
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项目类别:
-
资助金额:$24.39万
-
财政年份:1992
-
负责人:SHELDON W MAY
-
依托单位:
NEUROPEPTIDES--APPROACHES TO ALPHA-AMIDATION EFFECTORS
-
批准号:3298182
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项目类别:
-
资助金额:$21.15万
-
财政年份:1992
-
负责人:SHELDON W MAY
-
依托单位:
NEUROPEPTIDES--APPROACH TO AMIDATION EFFECTORS
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批准号:2684894
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项目类别:
-
资助金额:$20.79万
-
财政年份:1992
-
负责人:SHELDON W MAY
-
依托单位:
NEUROPEPTIDES--APPROACHES TO ALPHA-AMIDATION EFFECTORS
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批准号:3298181
-
项目类别:
-
资助金额:$22.66万
-
财政年份:1992
-
负责人:SHELDON W MAY
-
依托单位:
NEUROPEPTIDES--APPROACHES TO ALPHA-AMIDATION EFFECTORS
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批准号:2180417
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项目类别:
-
资助金额:$22.26万
-
财政年份:1992
-
负责人:SHELDON W MAY
-
依托单位:
NEUROPEPTIDES--APPROACH TO AMIDATION EFFECTORS
-
批准号:2900696
-
项目类别:
-
资助金额:$21.22万
-
财政年份:1992
-
负责人:SHELDON W MAY
-
依托单位:
NEUROPEPTIDES--APPROACHES TO ALPHA-AMIDATION EFFECTORS
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批准号:2180416
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项目类别:
-
资助金额:$21.02万
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财政年份:1992
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负责人:SHELDON W MAY
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依托单位:
METALLO MONOOXYGENASE CATALYSIS
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批准号:3284180
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项目类别:
-
资助金额:$3.37万
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财政年份:1987
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负责人:SHELDON W MAY
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依托单位:
METALLO MONOOXYGENASE CATALYSIS
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批准号:3284181
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项目类别:
-
资助金额:$10.65万
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财政年份:1985
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负责人:SHELDON W MAY
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依托单位:
METALLO MONOOXYGENASE CATALYSIS
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批准号:3284179
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项目类别:
-
资助金额:$10.92万
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财政年份:1985
-
负责人:SHELDON W MAY
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依托单位:
NON-HEME METALLO OXYGENASE CATALYSTS
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批准号:3271665
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项目类别:
-
资助金额:$16.97万
-
财政年份:1984
-
负责人:SHELDON W MAY
-
依托单位:
NON-HEME METALLO OXYGENASE CATALYSTS
-
批准号:3271664
-
项目类别:
-
资助金额:$16.2万
-
财政年份:1984
-
负责人:SHELDON W MAY
-
依托单位:
NON-HEME METALLO OXYGENASE CATALYSTS
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批准号:3271663
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项目类别:
-
资助金额:$15.41万
-
财政年份:1984
-
负责人:SHELDON W MAY
-
依托单位:
NOVEL ANTIHYPERTENSIVES: RATIONAL DESIGN AND EVALUATION
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批准号:3339577
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项目类别:
-
资助金额:$20.1万
-
财政年份:1982
-
负责人:SHELDON W MAY
-
依托单位:
NOVEL ANTIHYPERTENSIVES: RATIONAL DESIGN AND EVALUATION
-
批准号:3339576
-
项目类别:
-
资助金额:$24.86万
-
财政年份:1982
-
负责人:SHELDON W MAY
-
依托单位:
NOVEL ANTIHYPERTENSIVES: RATIONAL DESIGN AND EVALUATION
-
批准号:3339581
-
项目类别:
-
资助金额:$24.97万
-
财政年份:1982
-
负责人:SHELDON W MAY
-
依托单位:
NOVEL ANTIHYPERTENSIVES: RATIONAL DESIGN AND EVALUATION
-
批准号:3339580
-
项目类别:
-
资助金额:$24.48万
-
财政年份:1982
-
负责人:SHELDON W MAY
-
依托单位:
NOVEL ANTIHYPERTENSIVES: RATIONAL DESIGN AND EVALUATION
-
批准号:3339578
-
项目类别:
-
资助金额:$19.88万
-
财政年份:1982
-
负责人:SHELDON W MAY
-
依托单位:
NOVEL ANTIHYPERTENSIVES: RATIONAL DESIGN AND EVALUATION
-
批准号:3339575
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项目类别:
-
资助金额:$20.65万
-
财政年份:1982
-
负责人:SHELDON W MAY
-
依托单位:
NOVEL ANTIHYPERTENSIVES: RATIONAL DESIGN AND EVALUATION
-
批准号:3339579
-
项目类别:
-
资助金额:$20.75万
-
财政年份:1982
-
负责人:SHELDON W MAY
-
依托单位:
海外基金