ALPHA2 ADRENERGIC RECEPTOR DYSFUNCTION IN PATIENTS W/ REGIONAL LIPOAT
ALPHA2 ADRENERGIC RECEPTOR DYSFUNCTION IN PATIENTS W/ REGIONAL LIPOAT
批准号:
6264367
负责人:
CHARLES A STUART
金额:
$3.42万
依托单位国家:
美国
项目类别:
财政年份:
1998
资助国家:
美国
项目状态:
已结题
起止时间:
1998-12-01 至 1999-11-30
中文摘要
部分或全部脂肪萎缩的特征是胰岛素抵抗的糖尿病、高甘油三酯血症、肝脏脂肪浸润和高血压。这种综合征的病因尚不清楚。α2肾上腺素能受体是一种依赖GI的系统,通常主要在外周脂肪库中拮抗β肾上腺素能激动剂的脂解作用,并拮抗α1。
英文摘要
Partial or total lipoatrophy is characterized by insulin resistant diabetes, hypertiglyceridemia, fatty infiltration of the liver, and hypertension. The etiology of this syndrome is unknown. The alpha2 adrenergic receptor is a Gi-dependent system which normally antagonizes the lipolytic effects of beta adrenergic agonists primarily in peripheral fat depots and antagonizes alpha1.
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