Renal Clearable Organic Nanocarriers for Bioimaging and Drug Delivery.

Renal Clearable Organic Nanocarriers for Bioimaging and Drug Delivery.
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用于生物成像和药物递送的肾脏可透明有机纳米载体。

DOI:
10.1002/adma.201601101
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发表时间:
2016-10
期刊:
影响因子:
29.4
通讯作者:
Choi, Hak Soo
Choi, Hak Soo
中科院分区:
材料科学1区
文献类型:
--
作者:
Kang, Homan;Gravier, Julien;Bao, Kai;Wada, Hideyuki;Lee, Jeong Heon;Baek, Yoonji;El Fakhri, Georges;Gioux, Sylvain;Rubin, Brian P.;Coll, Jean-Luc;Choi, Hak Soo

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肾透明两性离子纳米载体(H-Dots)由用于电荷变化的ε-聚赖氨酸骨架、用于生物成像的近红外荧光团和用于潜在药物递送的β-环糊精组成。H-Dots显示出理想的体循环和快速分布,并在完全靶向肿瘤部位后通过肾排泄从正常组织/器官排出,而不被免疫系统非特异性摄取。
Renally cleared zwitterionic nanocarriers (H-Dots) are composed of ε-polylysine backbone for charge variations, near-infrared fluorophores for bioimaging, and β-cyclodextrins for potential drug delivery. H-Dots show ideal systemic circulation and rapid distribution and excrete from normal tissue/organ via renal excretion after complete targeting to the tumor site without nonspecific uptake by the immune system.
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